SCHEMBL30320628

SCHEMBL30320628

CC1(C)OB(c2ccc3c(c2)CCCC(=O)N3)OC1(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.46
PKM P14618 2/20 0.41
KIF11 P52732 4/20 0.40
IDO1 P14902 1/20 0.39
MAPK1 P28482 1/20 0.38
GSK3B P49841 1/20 0.37
BACE1 P56817 1/20 0.37
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
TBXAS1 P24557 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
LPL P06858 3/20 0.36
LIPG Q9Y5X9 3/20 0.36
PRMT5 O14744 1/20 0.35
WDR77 Q9BQA1 1/20 0.35
ROCK1 Q13464 1/20 0.35
NPC1 O15118 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28383719 1.00 MAPT (0.46) MAPTPKMKIF11IDO1MAPK1
SCHEMBL422134 0.92 PDE3B (0.44) MAPTPKMKIF11CYP1A2CYP2C9
SCHEMBL31243804 0.84 AHR (0.49) CYP1A2CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL454535 0.84 AHR (0.49) CYP1A2CYP11B1CYP11B2PDE3BPDE3A
SCHEMBL17042127 0.80 CA9 (0.50) BACE1CYP11B1CYP11B2LPLLIPG
SCHEMBL21382549 0.80 KDM4E (0.43) MAPTLPLLIPGROCK1CA1
SCHEMBL4158988 0.79 LPL (0.44) MAPK1BACE1LPLLIPGROCK1
SCHEMBL30284869 0.79 LPL (0.44) MAPK1BACE1LPLLIPGROCK1
SCHEMBL20612387 0.78 BRD9 (0.39) BACE1LPLLIPGPRMT5WDR77
SCHEMBL29984001 0.77 MAOB (0.47) MAPK1LPLLIPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4161936-A1 LPA RECEPTOR ANTAGONISTS AND USES THEREOF GILEAD SCIENCES, INC. (US) 2023-04-12 EP disclosed
CN-115867556-A LPA receptor antagonists and uses thereof 吉利德科学公司 2023-03-28 CN disclosed