SCHEMBL30338757

SCHEMBL30338757

NC(=O)c1nc(N2CCC(C(=O)O)CC2)ncc1F

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.51
CYP2C19 P33261 1/20 0.51
USP2 O75604 1/20 0.48
HPGD P15428 1/20 0.48
NPSR1 Q6W5P4 1/20 0.48
HSD17B10 Q99714 1/20 0.48
NEK2 P51955 6/20 0.44
TMPRSS15 P98073 2/20 0.41
ALDH1A1 P00352 1/20 0.41
NOTUM Q6P988 2/20 0.40
IDH2 P48735 1/20 0.40
SCN9A Q15858 1/20 0.40
PTPN11 Q06124 1/20 0.39
SYK P43405 1/20 0.39
ABL1 P00519 1/20 0.39
LMNA P02545 1/20 0.39
DYRK1A Q13627 1/20 0.38
AOC3 Q16853 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25294566 1.00 KDM4E (0.51) KDM4ECYP2C19USP2HPGDNPSR1
SCHEMBL30547531 0.84 KDM4E (0.55) KDM4ECYP2C19USP2HPGDNPSR1
SCHEMBL25253979 0.84 KDM4E (0.55) KDM4ECYP2C19USP2HPGDNPSR1
SCHEMBL20565681 0.83 KDM4E (0.56) KDM4ECYP2C19USP2HPGDNPSR1
Hydrochloric Acid SCHEMBL20565233 0.82 KDM4E (0.55) KDM4ECYP2C19USP2HPGDNPSR1
Trifluoroacetic Acid SCHEMBL30339273 0.82 KDM4E (0.49) KDM4ECYP2C19USP2HPGDNPSR1
SCHEMBL20565611 0.81 KDM4E (0.54) KDM4ECYP2C19USP2HPGDNPSR1
SCHEMBL20564608 0.79 KDM4E (0.51) KDM4ECYP2C19USP2HPGDNPSR1
SCHEMBL20165678 0.78 RIPK1 (0.67)
SCHEMBL20165680 0.78 RIPK1 (0.67)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116547281-A Isoxazolidines as RIPK1 inhibitors and uses thereof 赛诺菲 2023-08-04 CN disclosed
EP-4157835-A1 ISOXAZOLIDINES AS RIPK1 INHIBITORS AND USE THEREOF SANOFI (FR) 2023-04-05 EP disclosed