SCHEMBL30339587

SCHEMBL30339587

C=C(OC(=O)C(C)(C)Cn1nc(-c2ccccc2)c2c(C)cc(C)cc21)C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.34
PDE4A P27815 4/20 0.34
PDE4B Q07343 4/20 0.34
PDE4C Q08493 4/20 0.34
PDE4D Q08499 4/20 0.34
KMT2A Q03164 2/20 0.34
HTT P42858 2/20 0.34
MEN1 O00255 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
GAA P10253 1/20 0.33
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
POLB P06746 1/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
PTGDR2 Q9Y5Y4 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30339596 0.86 PTGER1 (0.41) THRBPDE4DKMT2AHTTMEN1
SCHEMBL30339630 0.85 KMT2A (0.37) PDE4APDE4BPDE4CPDE4DKMT2A
SCHEMBL30339960 0.84 MAPT (0.42) THRBKMT2AHTTMEN1GAA
SCHEMBL30339641 0.82 KMT2A (0.51) KMT2AHTTMEN1GAAALDH1A1
SCHEMBL30339514 0.80 MAPT (0.42) KMT2AHTTGAAALDH1A1KDM4E
SCHEMBL30339802 0.80 ALDH1A1 (0.45) KMT2AHTTMEN1GAAALDH1A1
SCHEMBL30339611 0.79 MAPT (0.46) KMT2AHTTMEN1GAAALDH1A1
SCHEMBL30339763 0.79 PTGER1 (0.44) KMT2AHTTGAAALDH1A1KDM4E
SCHEMBL30340291 0.79 MAPT (0.42) KMT2AHTTGAAALDH1A1KDM4E
SCHEMBL30339554 0.79 KDM4E (0.39) KMT2AHTTGAAALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116003326-A Synthesis method of trifluoromethyl indazole-containing derivative 河南师范大学 2023-04-25 CN disclosed