SCHEMBL30364591

SCHEMBL30364591

Cc1c(C)n(Cc2cccc(C(F)(F)F)c2)c2ccc(N)cc12

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PPARG P37231 9/20 0.54
PLA2G2A P14555 1/20 0.46
MAPT P10636 1/20 0.46
MAPK10 P53779 1/20 0.46
TP53 P04637 1/20 0.44
TAAR1 Q96RJ0 1/20 0.43
MAOB P27338 2/20 0.43
ALDH1A1 P00352 2/20 0.42
HPGD P15428 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23902746 1.00 PPARG (0.54) PPARGPLA2G2AMAPTMAPK10TP53
SCHEMBL30364951 0.80 PPARG (0.60) PPARG
SCHEMBL30364672 0.79 PPARG (0.45) PPARGMAPTMAPK10TP53TAAR1
SCHEMBL23902668 0.79 PPARG (0.45) PPARGMAPTMAPK10TP53TAAR1
Hydrochloric Acid SCHEMBL19896403 0.78 MAOB (0.50) MAPTMAPK10TAAR1MAOBALDH1A1
SCHEMBL23902707 0.78 ICMT (0.53) MAPTTP53TAAR1MAOBALDH1A1
SCHEMBL30364930 0.78 ICMT (0.53) MAPTTP53TAAR1MAOBALDH1A1
SCHEMBL23902644 0.76 PPARG (0.54) PPARGMAPT
SCHEMBL30241343 0.76 PPARG (0.54) PPARGMAPT
SCHEMBL28942976 0.74 ICMT (0.53) MAPTMAOBGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115667216-B (1H-indol-5-yl) acrylamide derivatives as inhibitors of TEAD proteins and HIPPO-YAP1/TAZ signaling cascades for the treatment of cancer 赛诺菲 2025-02-18 CN disclosed
CN-115667216-A (1H-indol-5-yl) acrylamide derivatives as TEAD proteins and inhibitors of the HIPPO-YAP1/TAZ signaling cascade for the treatment of cancer 赛诺菲 2023-01-31 CN disclosed