SCHEMBL30366459

SCHEMBL30366459

Cc1cccc(Oc2ccc(-c3c(-c4cnc(C#C[Si](C)(C)C(C)(C)C)cc4C)n(C)c4c(C#N)cnc(N)c34)cc2F)n1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
FGFR1 P11362 1/20 0.34
CYP2C9 P11712 1/20 0.34
FGFR2 P21802 1/20 0.34
FGFR4 P22455 1/20 0.34
FGFR3 P22607 1/20 0.34
CYP2C19 P33261 1/20 0.34
RET P07949 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30366887 0.91 CYP3A4 (0.41) ALOX5APFEN1CYP3A4CYP2D6FGFR1
SCHEMBL30366760 0.90 RET (0.32) RET
SCHEMBL30366837 0.89 ALOX5AP (0.36) ALOX5APFEN1CYP3A4CYP2D6FGFR1
SCHEMBL30366506 0.84 RET (0.32) ALOX5APFEN1RET
SCHEMBL28981129 0.82 ALOX5AP (0.33) ALOX5APFEN1CYP3A4CYP2D6FGFR1
SCHEMBL30366523 0.78 KDR (0.33) ALOX5APFEN1RET
SCHEMBL30325689 0.77 CYP3A4 (0.53) ALOX5APFEN1CYP3A4CYP2D6FGFR1
SCHEMBL22677138 0.75 CYP3A4 (0.49) ALOX5APFEN1CYP3A4CYP2D6FGFR1
SCHEMBL30303789 0.75 CYP3A4 (0.49) ALOX5APFEN1CYP3A4CYP2D6FGFR1
SCHEMBL30325855 0.75 CYP3A4 (0.53) ALOX5APFEN1CYP3A4CYP2D6FGFR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894481-A Nitrogen-containing heteroaryl compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-04-04 CN disclosed