SCHEMBL30366755

SCHEMBL30366755

COC(=O)c1cnc(Cl)c(I)c1N

nearest known ligand 0.42

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
GAA P10253 4/20 0.41
KDM4E B2RXH2 4/20 0.41
ALDH1A1 P00352 3/20 0.41
GLA P06280 2/20 0.41
ABL1 P00519 1/20 0.41
CFTR P13569 2/20 0.40
NQO2 P16083 6/20 0.40
MAPT P10636 2/20 0.40
HSD17B10 Q99714 2/20 0.39
POLB P06746 1/20 0.37
ATR Q13535 1/20 0.36
HPGD P15428 1/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28981135 1.00 TSHR (0.42) TSHRGAAKDM4EALDH1A1GLA
SCHEMBL7411789 0.85 TSHR (0.46) TSHRGAAKDM4EALDH1A1GLA
SCHEMBL23053815 0.83 TSHR (0.45) TSHRGAAKDM4EALDH1A1GLA
SCHEMBL31552179 0.83 NPC1 (0.48) KDM4EALDH1A1MAPTHSD17B10HPGD
SCHEMBL23043656 0.81 TSHR (0.42) TSHRGAAKDM4EALDH1A1GLA
SCHEMBL30391898 0.81 TSHR (0.42) TSHRGAAKDM4EALDH1A1GLA
SCHEMBL25239223 0.77 TSHR (0.42) TSHRGAAKDM4EALDH1A1GLA
SCHEMBL31140734 0.77 TSHR (0.42) TSHRGAAKDM4EALDH1A1GLA
SCHEMBL31523457 0.76 MAPT (0.39) TSHRGAAKDM4EALDH1A1GLA
SCHEMBL19134228 0.75 TSHR (0.46) TSHRGAAKDM4EALDH1A1GLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115894481-A Nitrogen-containing heteroaryl compound, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2023-04-04 CN disclosed