SCHEMBL25239223

SCHEMBL25239223

COC(=O)c1cnc(N)c(I)c1Cl

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.42
GAA P10253 4/20 0.41
ALDH1A1 P00352 4/20 0.41
KDM4E B2RXH2 4/20 0.41
GLA P06280 2/20 0.41
ABL1 P00519 1/20 0.41
MAPT P10636 2/20 0.40
NQO2 P16083 7/20 0.39
CFTR P13569 2/20 0.39
HSD17B10 Q99714 2/20 0.39
HPGD P15428 2/20 0.36
CASP1 P29466 1/20 0.36
CASP7 P55210 1/20 0.36
ATM Q13315 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31140734 1.00 TSHR (0.42) TSHRGAAALDH1A1KDM4EGLA
SCHEMBL25784214 0.82 TSHR (0.44) TSHRGAAALDH1A1KDM4EGLA
SCHEMBL2650690 0.82 SMN1; SMN2 (0.40) TSHRGAAALDH1A1KDM4EGLA
SCHEMBL31140761 0.81 TSHR (0.42) TSHRGAAALDH1A1KDM4EGLA
SCHEMBL5254344 0.81 KDM4E (0.44) TSHRGAAALDH1A1KDM4EGLA
SCHEMBL25289336 0.81 TSHR (0.42) TSHRGAAALDH1A1KDM4EGLA
SCHEMBL31140730 0.80 NNMT (0.44) TSHR
SCHEMBL25284307 0.80 NNMT (0.44) TSHR
SCHEMBL28981135 0.77 TSHR (0.42) TSHRGAAALDH1A1KDM4EGLA
SCHEMBL30366755 0.77 TSHR (0.42) TSHRGAAALDH1A1KDM4EGLA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116779-A1 DIALKYNE COMPOUND AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-06-29 WO disclosed
WO-2023116779-A1 DIALKYNE COMPOUND AND USE THEREOF 上海艾力斯医药科技股份有限公司 2023-06-29 WO disclosed