SCHEMBL30367066

SCHEMBL30367066

C[C@H](N)c1cccc(C(F)F)c1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2D6 P10635 1/20 0.45
NFKB1 P19838 1/20 0.45
PNMT P11086 1/20 0.45
LMNA P02545 3/20 0.44
ALDH1A1 P00352 1/20 0.44
GLA P06280 1/20 0.44
PDE2A O00408 1/20 0.36
KRAS P01116 1/20 0.36
SOS1 Q07889 1/20 0.36
CFD P00746 1/20 0.34
SLC6A2 P23975 2/20 0.33
FAAH O00519 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
GABRA1 P14867 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33
GABRB1 P18505 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23326566 1.00 CYP1A2 (0.45) CYP1A2CYP3A4CYP2D6NFKB1PNMT
SCHEMBL30577965 1.00 CYP1A2 (0.45) CYP1A2CYP3A4CYP2D6NFKB1PNMT
SCHEMBL29672766 1.00 CYP1A2 (0.45) CYP1A2CYP3A4CYP2D6NFKB1PNMT
SCHEMBL21132678 1.00 CYP1A2 (0.45) CYP1A2CYP3A4CYP2D6NFKB1PNMT
SCHEMBL27089982 1.00 CYP1A2 (0.45) CYP1A2CYP3A4CYP2D6NFKB1PNMT
Hydrochloric Acid SCHEMBL23247765 0.98 LMNA (0.47) CYP1A2CYP3A4CYP2D6NFKB1PNMT
Hydrochloric Acid SCHEMBL29180804 0.98 LMNA (0.47) CYP1A2CYP3A4CYP2D6NFKB1PNMT
Hydrochloric Acid SCHEMBL23247764 0.98 LMNA (0.47) CYP1A2CYP3A4CYP2D6NFKB1PNMT
Hydrochloric Acid SCHEMBL29755142 0.98 LMNA (0.47) CYP1A2CYP3A4CYP2D6NFKB1PNMT
Hydrochloric Acid SCHEMBL29901777 0.98 LMNA (0.47) CYP1A2CYP3A4CYP2D6NFKB1PNMT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117396472-A SOS1 inhibitors and uses thereof 上海齐鲁锐格医药研发有限公司 2024-01-12 CN disclosed
CN-116082360-A Polycyclic compounds as SOS1 inhibitors 昆药集团股份有限公司 2023-05-09 CN disclosed