SCHEMBL30367208

SCHEMBL30367208

CC(C)C(=O)N1CC=C(c2nc(-c3ccc(N)cc3)c3c(N)nccn23)CC1

nearest known ligand 0.60

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TNK2 Q07912 12/20 0.60
BTK Q06187 4/20 0.47
EGFR P00533 2/20 0.43
TEC P42680 2/20 0.43
TXK P42681 2/20 0.43
BMX P51813 2/20 0.43
ITK Q08881 2/20 0.43
NAMPT P43490 3/20 0.41
GRIA1 P42261 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29721103 0.77 BTK (0.73) TNK2BTK
SCHEMBL4361853 0.75 TNK2 (1.00) TNK2BTK
SCHEMBL399045 0.73 IGF1R (0.62) TNK2EGFR
SCHEMBL6940080 0.70 RAF1 (0.67) TNK2BTKEGFR
SCHEMBL27678612 0.70 IGF1R (0.59) TNK2EGFR
SCHEMBL13504841 0.69 TNK2 (0.78) TNK2BTK
SCHEMBL11980652 0.69 RAF1 (0.54) TNK2EGFR
SCHEMBL6942526 0.68 PIK3CA (0.55) TNK2BTKEGFR
SCHEMBL3897506 0.68 IGF1R (0.57) TNK2EGFR
SCHEMBL30367439 0.67 BTK (0.50) BTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116437918-A Pyrazolopyridine compounds as TAM inhibitors 上海德琪医药科技有限公司 2023-07-14 CN disclosed
WO-2023051464-A1 PYRAZOLOPYRIDINE COMPOUNDS AS TAM INHIBITORS SHANGHAI ANTENGENE CORPORATION LIMITED (CN) 2023-04-06 WO disclosed