SCHEMBL30375783

SCHEMBL30375783

C[C@@H](NC(=O)c1ccc2c(c1)CC(=O)N2)c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 12/20 0.65
IMPDH2 P12268 2/20 0.52
ALDH1A1 P00352 2/20 0.51
NPC1 O15118 1/20 0.51
LMNA P02545 1/20 0.51
ANPEP P15144 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25315485 1.00 SMYD3 (0.65) SMYD3IMPDH2ALDH1A1NPC1LMNA
SCHEMBL30376200 1.00 SMYD3 (0.65) SMYD3IMPDH2ALDH1A1NPC1LMNA
SCHEMBL18006588 1.00 SMYD3 (0.65) SMYD3IMPDH2ALDH1A1NPC1LMNA
SCHEMBL18006574 0.90 SMYD3 (0.53) SMYD3IMPDH2ALDH1A1NPC1LMNA
SCHEMBL25312585 0.89 SMYD3 (0.55) SMYD3ANPEP
SCHEMBL25312590 0.89 SMYD3 (0.55) SMYD3ANPEP
SCHEMBL30376271 0.89 SMYD3 (0.55) SMYD3ANPEP
SCHEMBL25311225 0.88 SMYD3 (0.52) SMYD3ANPEP
SCHEMBL25313541 0.88 AKT1 (0.56) SMYD3ANPEP
SCHEMBL25311973 0.88 SMYD3 (0.62) SMYD3ALDH1A1ANPEP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4157858-A2 SMALL MOLECULE INHIBITORS OF GRK5 AND GRK5 SUBFAMILY MEMBERS AND USES THEREOF The Regents of The University of Michigan (US) 2023-04-05 EP disclosed