SCHEMBL3038071

SCHEMBL3038071

COc1cc(-c2cc3cc(N)ccc3[nH]2)c2c(c1OS(C)(=O)=O)CNC2=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 10/20 0.46
KDR P35968 10/20 0.46
NQO2 P16083 1/20 0.39
CDK1 P06493 1/20 0.39
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
RAB9A P51151 1/20 0.34
KMT2A Q03164 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CA2 P00918 2/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA9 Q16790 1/20 0.32
CHEK1 O14757 2/20 0.31
WEE1 P30291 2/20 0.31
CYP2A6 P11509 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL3048315 0.99 AURKA (0.45) AURKAKDRNQO2CDK1KDM4E
SCHEMBL3043839 0.89 KDR (0.46) AURKAKDRNQO2CDK1KDM4E
SCHEMBL3047326 0.89 AURKA (0.53) AURKAKDRNQO2CDK1KDM4E
Hydrochloric Acid SCHEMBL3042483 0.87 AURKA (0.43) AURKAKDRNQO2CDK1KDM4E
Hydrochloric Acid SCHEMBL3047981 0.87 KDR (0.50) AURKAKDRNQO2CDK1KDM4E
SCHEMBL3052415 0.86 KDR (0.43) AURKAKDRNQO2CDK1KDM4E
SCHEMBL3045069 0.85 AURKA (0.42) AURKAKDRNQO2CDK1KDM4E
SCHEMBL3054784 0.85 AURKA (0.42) AURKAKDRNQO2CDK1KDM4E
SCHEMBL3046942 0.85 AURKA (0.44) AURKAKDRNQO2CDK1KDM4E
Hydrochloric Acid SCHEMBL3049923 0.84 AURKA (0.42) AURKAKDRNQO2CDK1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9018209-B2 Compounds and methods for the treatment of viruses and cancer YALE UNIVERSITY (US) 2015-04-28 US disclosed
US-20100222352-A1 Compounds and Methods for the Treatment of Viruses and Cancer YALE UNIVERSITY (US) 2010-09-02 US disclosed
US-7745641-B2 Nitrogen-containing heterocyclic compound KYOWA HAKKO KIRIN CO., LTD. (JP) 2010-06-29 US disclosed
US-20090054407-A1 Nitrogen-containing heterocyclic compound KYOWA HAKKO KOGYO CO., LTD. (JP) 2009-02-26 US disclosed
EP-1880993-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUND KYOWA HAKKO KOGYO CO., LTD. (JP) 2008-01-23 EP disclosed
WO-2007038387-A2 COMPOUNDS AND METHODS FOR THE TREATMENT OF VIRUSES AND CANCER YALE UNIVERSITY (US) 2007-04-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090054407-A1 Nitrogen-containing heterocyclic compound NR4A1, NR5A2, PRMT8 AURKA 2312/4885KDR 3226/4885NQO2 308/4885
US-20100222352-A1 Compounds and Methods for the Treatment of Viruses and Cancer RCOR1, RCOR3, CCNT1 AURKA 3222/4885KDR 1458/4885NQO2 1956/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.