SCHEMBL30384259

SCHEMBL30384259

COc1cccc(C=CC(=O)c2ccccc2O)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 8/20 1.00
MAOA P21397 3/20 1.00
NR1H4 Q96RI1 3/20 0.82
ABCG2 Q9UNQ0 5/20 0.80
CYP2D6 P10635 2/20 0.72
CYP2C9 P11712 2/20 0.72
CYP2C19 P33261 2/20 0.72
MAPT P10636 2/20 0.72
CASP3 P42574 1/20 0.72
SENP8 Q96LD8 1/20 0.72
SENP7 Q9BQF6 1/20 0.72
SENP6 Q9GZR1 1/20 0.72
CYP1A2 P05177 1/20 0.72
CYP3A4 P08684 1/20 0.72
HSP90AA1 P07900 1/20 0.72
NPC1 O15118 1/20 0.69
LMNA P02545 1/20 0.69
RECQL P46063 1/20 0.69
RAB9A P51151 1/20 0.69
ATM Q13315 1/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25225627 1.00 MAOB (1.00) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL5085597 1.00 MAOB (1.00) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL5085601 1.00 MAOB (1.00) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL31233034 0.89 ABCG2 (1.00) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL5138658 0.89 ABCG2 (1.00) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL5138657 0.89 ABCG2 (1.00) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL7196541 0.89 MAOB (0.80) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL7196545 0.89 MAOB (0.80) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL31234600 0.89 MAOB (0.80) MAOBMAOANR1H4ABCG2CYP2D6
SCHEMBL25202062 0.88 MAOB (1.00) MAOBMAOANR1H4ABCG2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4429763-A1 COMPOSITIONS AND METHODS FOR TREATING BLEEDING AND BLEEDING DISORDERS Yewsavin, Inc. (US) 2024-09-18 EP disclosed
WO-2023086388-A1 COMPOSITIONS AND METHODS FOR TREATING BLEEDING AND BLEEDING DISORDERS YewSavin, Inc. (US) 2023-05-19 WO disclosed