SCHEMBL30388409

SCHEMBL30388409

N#Cc1cc2c(cc1NC(=O)c1ccccc1)OCO2

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 9/20 0.65
RAB9A P51151 9/20 0.65
KMT2A Q03164 3/20 0.55
PTGS2 P35354 1/20 0.55
SMN1; SMN2 Q16637 6/20 0.52
ALDH1A1 P00352 5/20 0.52
MAPT P10636 5/20 0.52
KDM4E B2RXH2 2/20 0.52
NPSR1 Q6W5P4 2/20 0.52
TDP1 Q9NUW8 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MEN1 O00255 2/20 0.51
POLB P06746 1/20 0.51
PKM P14618 2/20 0.50
HPGD P15428 3/20 0.49
LMNA P02545 1/20 0.49
GAA P10253 1/20 0.48
THRB P10828 1/20 0.47
TP53 P04637 1/20 0.47
CYP1A2 P05177 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1623124 0.90 NPC1 (0.54) NPC1RAB9AKMT2APTGS2SMN1; SMN2
SCHEMBL11785020 0.78 TP53 (0.73) NPC1RAB9APTGS2SMN1; SMN2ALDH1A1
SCHEMBL30388616 0.77 NPC1 (0.58) NPC1RAB9AKMT2APTGS2SMN1; SMN2
SCHEMBL1343798 0.75 KDM4E (0.63) NPC1RAB9AKMT2ASMN1; SMN2ALDH1A1
SCHEMBL21366573 0.74 NPC1 (0.54) NPC1RAB9AKMT2APTGS2SMN1; SMN2
SCHEMBL23048315 0.73 KCNMA1 (0.64) NPC1RAB9AKMT2ASMN1; SMN2ALDH1A1
SCHEMBL18154023 0.73 HDAC1 (0.62) NPC1RAB9AKMT2ASMN1; SMN2MAPT
SCHEMBL3530485 0.73 MAPT (0.62) NPC1RAB9AKMT2ASMN1; SMN2MAPT
SCHEMBL400049 0.73 KCNMA1 (0.64) NPC1RAB9AKMT2ASMN1; SMN2ALDH1A1
SCHEMBL13102688 0.73 KCNMA1 (0.60) NPC1RAB9AKMT2ASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3596067-B1 PYRAZOLE DERIVATIVES FOR THE TREATMENT OF CYSTIC FIBROSIS FONDAZIONE ST ITALIANO TECNOLOGIA (IT) 2023-06-07 EP claimed