SCHEMBL30397404

SCHEMBL30397404

CC(C)Oc1ncn([C@@H]2CCC[C@@H](Nc3ncc(C(F)(F)F)c(OC4COC4)n3)C2)n1

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ULK1 O75385 1/20 0.39
CDK2 P24941 10/20 0.36
KDR P35968 2/20 0.36
CCNE1 P24864 8/20 0.35
PTK2 Q05397 1/20 0.35
CDK1 P06493 5/20 0.34
CCNB1 P14635 2/20 0.34
CDK4 P11802 1/20 0.33
CCND1 P24385 1/20 0.33
CCND3 P30281 1/20 0.33
CDK6 Q00534 1/20 0.33
CCNT1 O60563 3/20 0.33
CCNK O75909 3/20 0.33
CDK9 P50750 3/20 0.33
CDK12 Q9NYV4 3/20 0.33
LRRK2 Q5S007 4/20 0.32
CYP1A2 P05177 1/20 0.32
MAPK3 P27361 1/20 0.32
HSD11B1 P28845 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30396062 1.00 ULK1 (0.39) ULK1CDK2KDRCCNE1PTK2
SCHEMBL30397887 1.00 ULK1 (0.39) ULK1CDK2KDRCCNE1PTK2
SCHEMBL30398079 1.00 ULK1 (0.39) ULK1CDK2KDRCCNE1PTK2
SCHEMBL30397421 0.93 ULK1 (0.39) ULK1CDK2KDRCCNE1PTK2
SCHEMBL30397769 0.93 ULK1 (0.39) ULK1CDK2KDRCCNE1PTK2
SCHEMBL25418204 0.93 ULK1 (0.39) ULK1CDK2KDRCCNE1PTK2
SCHEMBL30397668 0.93 ULK1 (0.39) ULK1CDK2KDRCCNE1PTK2
SCHEMBL30397015 0.93 ULK1 (0.39) ULK1CDK2KDRCCNE1PTK2
SCHEMBL30397251 0.91 ULK1 (0.41) ULK1CDK2KDRCCNE1PTK2
SCHEMBL30398072 0.91 ULK1 (0.41) ULK1CDK2KDRCCNE1PTK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023091726-A1 INHIBITORS OF CYCLIN‑DEPENDENT KINASE 12 (CDK12) SYROS PHARMACEUTICALS, INC. (US) 2023-05-25 WO disclosed