Aptiganel

Aptiganel

SCHEMBL30416816

CCc1cccc(N(C)/C(N)=N/c2cccc3ccccc23)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 13/20 1.00
TP53 P04637 1/20 1.00
CYP2D6 P10635 1/20 1.00
TSHR P16473 1/20 1.00
THPO P40225 1/20 1.00
MTOR P42345 1/20 1.00
MEN1 O00255 1/20 0.98
LMNA P02545 1/20 0.98
MAPT P10636 1/20 0.98
PMP22 Q01453 1/20 0.98
KMT2A Q03164 1/20 0.98
TDP1 Q9NUW8 1/20 0.98

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Aptiganel SCHEMBL30481113 1.00 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
Aptiganel SCHEMBL21775476 1.00 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
Aptiganel SCHEMBL151145 1.00 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
Aptiganel SCHEMBL7414862 0.99 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6719553 0.86 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6727461 0.84 SIGMAR1 (0.73) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6719522 0.84 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL16887967 0.83 SIGMAR1 (0.71) SIGMAR1TP53CYP2D6TSHRTHPO
Hydrochloric Acid SCHEMBL7412867 0.82 SIGMAR1 (0.97) SIGMAR1TP53CYP2D6TSHRTHPO
SCHEMBL6728156 0.81 SIGMAR1 (1.00) SIGMAR1TP53CYP2D6TSHRTHPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110831584-B Targeted drug rescue with novel compositions, combinations and methods thereof 埃克塞瓦有限责任公司 2023-03-10 CN claimed
CN-110831584-B Targeted drug rescue with novel compositions, combinations and methods thereof 埃克塞瓦有限责任公司 2023-03-10 CN disclosed