SCHEMBL30417469

SCHEMBL30417469

Cc1cccc2c(=O)[nH]c(CCN3CCC[C@@H]3CO)cc12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 3/20 1.00
CCNE2 O96020 1/20 0.43
CDK4 P11802 1/20 0.43
PRKACA P17612 1/20 0.43
PRKACG P22612 1/20 0.43
PRKACB P22694 1/20 0.43
CCND1 P24385 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
CAMK2B Q13554 1/20 0.43
CAMK2G Q13555 1/20 0.43
CAMK2D Q13557 1/20 0.43
CAMK2A Q9UQM7 1/20 0.43
SPHK2 Q9NRA0 2/20 0.42
SPHK1 Q9NYA1 2/20 0.42
HRH3 Q9Y5N1 2/20 0.42
TNKS O95271 6/20 0.40
KDM4E B2RXH2 2/20 0.40
HTR1D P28221 1/20 0.39
HTR1B P28222 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1945766 1.00 PARP1 (1.00) PARP1CCNE2CDK4PRKACAPRKACG
SCHEMBL30090665 1.00 PARP1 (1.00) PARP1CCNE2CDK4PRKACAPRKACG
SCHEMBL1946020 1.00 PARP1 (1.00) PARP1CCNE2CDK4PRKACAPRKACG
SCHEMBL3443321 1.00 PARP1 (1.00) PARP1CCNE2CDK4PRKACAPRKACG
Hydrochloric Acid SCHEMBL1946668 0.99 PARP1 (0.98) PARP1CCNE2CDK4PRKACAPRKACG
Bromide SCHEMBL1944264 0.99 PARP1 (0.98) PARP1CCNE2CDK4PRKACAPRKACG
Bromide SCHEMBL1944266 0.99 PARP1 (0.98) PARP1CCNE2CDK4PRKACAPRKACG
Hydrochloric Acid SCHEMBL1946669 0.99 PARP1 (0.98) PARP1CCNE2CDK4PRKACAPRKACG
Bromide SCHEMBL1946605 0.98 PARP1 (0.96) PARP1CCNE2CDK4PRKACAPRKACG
Bromide SCHEMBL1946607 0.98 PARP1 (0.96) PARP1CCNE2CDK4PRKACAPRKACG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4419094-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF HYPERPROLIFERATIVE, INFLAMMATORY, AND IMMUNOLOGICAL DISEASES, AND INFECTIONS Edison Oncology (US) 2024-08-28 EP disclosed
WO-2023069727-A1 COMPOSITIONS AND METHODS FOR TREATMENT OF HYPERPROLIFERATIVE, INFLAMMATORY, AND IMMUNOLOGICAL DISEASES, AND INFECTIONS EDISON ONCOLOGY (US) 2023-04-27 WO disclosed