SCHEMBL30419263

SCHEMBL30419263

Cc1cncc(C(=O)NC2CCN(C)CC2)c1

nearest known ligand 0.69

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 6/20 0.69
SSTR5 P35346 14/20 0.58
SSTR1 P30872 1/20 0.53
HRH1 P35367 1/20 0.53
KCNH2 Q12809 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15366968 0.85 SMYD3 (0.67) SMYD3
SCHEMBL16415945 0.83 ALDH1A1 (0.53) SMYD3
SCHEMBL19133764 0.82 HDAC4 (0.47) SMYD3
SCHEMBL30419625 0.82 SMYD3 (1.00) SMYD3SSTR5
SCHEMBL21489983 0.82 SMYD3 (1.00) SMYD3SSTR5
SCHEMBL2964004 0.82 SMYD3 (0.71) SMYD3SSTR5SSTR1HRH1
SCHEMBL19701356 0.82 SMYD3 (1.00) SMYD3SSTR5
SCHEMBL27704323 0.81 SMYD3 (0.59) SMYD3SSTR5SSTR1HRH1KCNH2
SCHEMBL2953693 0.80 SMYD3 (0.58) SMYD3SSTR5SSTR1HRH1
SCHEMBL2957930 0.80 SSTR5 (0.72) SSTR5SSTR1HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240299352-A1 COMBINATION THERAPIES WITH SETD2 INHIBITORS Epizyme, Inc. 2024-09-12 US disclosed
US-20230133671-A1 SETD2 INHIBITORS AND RELATED METHODS AND USES, INCLUDING COMBINATION THERAPIES Epizyme, Inc. (US) 2023-05-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240299352-A1 COMBINATION THERAPIES WITH SETD2 INHIBITORS SETD2, CARM1, SETDB1 SMYD3 386/4885SSTR5 4085/4885SSTR1 3938/4885
US-20230133671-A1 SETD2 INHIBITORS AND RELATED METHODS AND USES, INCLUDING COMBINATION THERAPIES EZH2, HDAC2, SETD2 SMYD3 489/4885SSTR5 4008/4885SSTR1 4332/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.