SCHEMBL30420643

SCHEMBL30420643

Cc1noc(C)c1-c1ccc(N)nc1F

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 9/20 0.42
BRD2 P25440 1/20 0.42
MBOAT4 Q96T53 1/20 0.40
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
AR P10275 1/20 0.38
BTK Q06187 1/20 0.38
JAK2 O60674 1/20 0.38
CYP1A2 P05177 4/20 0.37
CYP3A4 P08684 4/20 0.37
HSD17B10 Q99714 3/20 0.37
CYP2C19 P33261 2/20 0.37
LMNA P02545 1/20 0.37
TSHR P16473 1/20 0.37
CLK4 Q9HAZ1 1/20 0.37
USP2 O75604 1/20 0.37
ALOX15 P16050 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24103788 1.00 BRD4 (0.42) BRD4BRD2MBOAT4NPC1POLB
SCHEMBL30522525 0.74 MAP4K4 (0.43) BRD4BRD2MBOAT4NPC1POLB
SCHEMBL15206943 0.72 BRD4 (0.44) BRD4BRD2MBOAT4CYP1A2CYP3A4
SCHEMBL18249941 0.71 FFAR1 (0.43) BRD4BRD2NPC1POLBCASP3
SCHEMBL16404611 0.69 BRD4 (0.56) BRD4BRD2NPC1POLBCASP3
SCHEMBL12362771 0.69 BRD4 (0.49) BRD4BRD2ARBTKCYP1A2
SCHEMBL19754246 0.68 BRD4 (0.46) BRD4BRD2MBOAT4NPC1POLB
SCHEMBL29836739 0.68 BRD4 (0.46) BRD4BRD2MBOAT4ARJAK2
SCHEMBL27321340 0.67 KDM4E (0.36) NOS3NOS1NOS2
SCHEMBL13036090 0.67 NPC1 (0.47) BRD4BRD2NPC1POLBCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116209664-A Small molecule modulators of IL-17 利奥制药有限公司 2023-06-02 CN disclosed