SCHEMBL30430643

SCHEMBL30430643

[2H]C1([2H])OC(=O)c2c(Br)cccc21

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA7 P43166 1/20 0.34
CA9 Q16790 1/20 0.34
PARP1 P09874 1/20 0.32
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
PIM1 P11309 1/20 0.31
CSNK1A1 P48729 1/20 0.31
CDK5 Q00535 1/20 0.31
ROCK1 Q13464 1/20 0.31
DYRK1A Q13627 1/20 0.31
LRRK2 Q5S007 1/20 0.31
CLK4 Q9HAZ1 1/20 0.31
DYRK1B Q9Y463 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
TYMS P04818 1/20 0.31
CYP1A2 P05177 1/20 0.31
HPGD P15428 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL855553 0.80 MAOA (0.47) CA1CA2CA7CA9PARP1
SCHEMBL17397682 0.67 KDM4E (0.37) CA1CA2CA7CA9PARP1
SCHEMBL1150797 0.65 KDM4E (0.38) CA1CA2CA7CA9PARP1
SCHEMBL28494219 0.65 CA1 (0.34) CA1CA2CA7CA9PARP1
SCHEMBL12213268 0.65 CYP3A4 (0.43) CA1CA2CA7CA9PARP1
SCHEMBL3046612 0.63 AURKA (0.57) CA1CA2CA7CA9PARP1
SCHEMBL13151641 0.63 MAOA (0.32) MAOAMAOBKDM4EALDH1A1TYMS
SCHEMBL5238902 0.63 MAOA (0.48) CA1CA2CA7CA9MAOA
SCHEMBL12430518 0.63 MAOA (0.44) CA1CA2CA7CA9MAOA
SCHEMBL1768468 0.62 AHR (0.43) CA1CA2CA7CA9PARP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023044171-A1 INHIBITORS OF CYSTEINE PROTEASES AND METHODS OF USE THEREOF Pardes Biosciences, Inc. (US) 2023-03-23 WO disclosed