SCHEMBL30435151

SCHEMBL30435151

CC(C)NC(=O)NCc1ccc(C(F)(F)F)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 2/20 0.57
NAMPT P43490 2/20 0.54
LSS P48449 1/20 0.52
EPHX2 P34913 2/20 0.50
PPARG P37231 2/20 0.50
TSHR P16473 2/20 0.50
MAPK1 P28482 1/20 0.50
PPARA Q07869 1/20 0.50
OPRM1 P35372 1/20 0.49
OPRL1 P41146 1/20 0.49
HDAC3 O15379 1/20 0.49
HDAC1 Q13547 1/20 0.49
HDAC2 Q92769 1/20 0.49
HDAC10 Q969S8 1/20 0.49
HDAC11 Q96DB2 1/20 0.49
HDAC8 Q9BY41 1/20 0.49
HDAC6 Q9UBN7 1/20 0.49
ALDH1A1 P00352 1/20 0.49
MEN1 O00255 1/20 0.48
GAA P10253 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24575984 0.85 MTOR (0.69) MTORNAMPTLSSOPRM1OPRL1
SCHEMBL12375168 0.82 MAPK1 (0.70) TSHRMAPK1ALDH1A1MEN1GAA
SCHEMBL12757446 0.81 ERCC1 (0.55) MTORNAMPTLSSEPHX2PPARG
SCHEMBL21202238 0.79 TGM2 (0.51) TSHRMAPK1ALDH1A1MEN1GAA
SCHEMBL24568690 0.79 NAMPT (0.66) NAMPTMAPK1ALDH1A1
SCHEMBL12375169 0.79 TSHR (0.70) LSSEPHX2TSHRALDH1A1MEN1
SCHEMBL12252067 0.78 MAPT (0.69) ALDH1A1MEN1KMT2AANPEP
SCHEMBL2629356 0.78 LSS (0.59) MTORNAMPTLSSEPHX2PPARG
SCHEMBL22522168 0.78 LSS (0.52) MTORNAMPTLSSEPHX2PPARG
SCHEMBL3879096 0.78 PPARA (0.56) MTORNAMPTLSSEPHX2PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4185296-A1 ADENOSINE A2A AND A2B RECEPTOR DUAL ANTAGONISTS FOR IMMUNO-ONCOLOGY Merck Sharp & Dohme LLC (US) 2023-05-31 EP disclosed