SCHEMBL30438589

SCHEMBL30438589

CNCCC(OCc1cccc(NC(=O)c2cnc(OC)nc2)c1)c1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 19/20 0.51
SLC6A2 P23975 11/20 0.51
SLC1A3 P43003 1/20 0.45
SLC1A2 P43004 1/20 0.45
SLC1A1 P43005 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20917135 1.00 CACNA2D1 (0.51) CACNA2D1SLC6A2SLC1A3SLC1A2SLC1A1
SCHEMBL20917088 0.88 CACNA2D1 (0.52) CACNA2D1SLC6A2
SCHEMBL20917105 0.88 CACNA2D1 (0.49) CACNA2D1SLC6A2SLC1A2SLC1A1
SCHEMBL20917044 0.88 CACNA2D1 (0.51) CACNA2D1SLC6A2SLC1A3SLC1A2SLC1A1
SCHEMBL20917077 0.84 KCNK3 (0.54) CACNA2D1
SCHEMBL20917140 0.83 CACNA2D1 (0.50) CACNA2D1SLC6A2
SCHEMBL20917082 0.82 CACNA2D1 (0.50) CACNA2D1SLC6A2
SCHEMBL30438634 0.82 CACNA2D1 (0.50) CACNA2D1SLC6A2
SCHEMBL21349106 0.76 TAS1R3 (0.56)
SCHEMBL20917092 0.76 CACNA2D1 (0.56) CACNA2D1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111225901-B Propylamine derivatives for the treatment of pain and pain-related disorders 埃斯特韦制药股份公司 2023-07-04 CN claimed
CN-111225901-B Propylamine derivatives for the treatment of pain and pain-related disorders 埃斯特韦制药股份公司 2023-07-04 CN disclosed