SCHEMBL30449333

SCHEMBL30449333

COc1ccc(COc2cccc(NS(C)(=O)=O)c2Br)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 8/20 0.56
NR3C1 P04150 1/20 0.48
HTR1A P08908 1/20 0.47
ADRA1D P25100 1/20 0.47
ADRA1A P35348 1/20 0.47
ADRA1B P35368 1/20 0.47
HDAC3 O15379 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC2 Q92769 1/20 0.45
NCOR2 Q9Y618 1/20 0.45
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
AR P10275 1/20 0.45
HPGD P15428 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
ABCB1 P08183 2/20 0.43
SMPD1 P17405 1/20 0.43
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8605381 0.87 CYP19A1 (0.54) CYP19A1NR3C1NPC1RAB9AAR
SCHEMBL30448631 0.81 CYP19A1 (0.66) CYP19A1NR3C1HTR1AADRA1DADRA1A
SCHEMBL21824613 0.78 NPC1 (0.55) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL22989897 0.74 MAOB (0.51) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL5203042 0.74 CYP19A1 (0.64) CYP19A1NR3C1HTR1AADRA1DADRA1A
SCHEMBL3446415 0.74 ALDH1A1 (0.54) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL3447303 0.72 ABCB1 (0.55) HTR1AADRA1DADRA1AADRA1BNPC1
SCHEMBL621125 0.71 NPC1 (0.50) CYP19A1HTR1AADRA1DADRA1AADRA1B
SCHEMBL3296630 0.71 CYP19A1 (1.00) CYP19A1
SCHEMBL22440563 0.71 NPC1 (0.53) HTR1AADRA1DADRA1AADRA1BNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332948-A Nitrogen-containing tetracyclic compound, preparation method and medicinal application thereof 翰森生物有限责任公司 2023-06-27 CN disclosed