SCHEMBL30450950

SCHEMBL30450950

COc1cc(-c2ncncc2-c2ccc(SC)cc2)cc(OC)c1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.60
KMT2A Q03164 1/20 0.45
CYP1A1 P04798 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP1B1 Q16678 1/20 0.45
BRD4 O60885 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
LMNA P02545 1/20 0.41
HTT P42858 1/20 0.41
NCOA1 Q15788 1/20 0.41
NCOA3 Q9Y6Q9 1/20 0.41
CHEK2 O96017 1/20 0.41
FYN P06241 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29015021 1.00 KCNH2 (0.60) KCNH2KMT2ACYP1A1CYP1A2CYP1B1
SCHEMBL29014986 0.86 KCNH2 (0.62) KCNH2KMT2ABRD4NPSR1LMNA
SCHEMBL30450307 0.86 KCNH2 (0.62) KCNH2KMT2ABRD4NPSR1LMNA
SCHEMBL29014967 0.85 KCNH2 (0.63) KCNH2KMT2ANPSR1LMNAHTT
SCHEMBL30451554 0.85 KCNH2 (0.63) KCNH2KMT2ANPSR1LMNAHTT
SCHEMBL30451069 0.84 KCNH2 (0.62) KCNH2KMT2ABRD4NPSR1LMNA
SCHEMBL29014998 0.84 KCNH2 (0.62) KCNH2KMT2ABRD4NPSR1LMNA
SCHEMBL29015012 0.81 KCNH2 (0.71) KCNH2KMT2ANPSR1LMNAHTT
SCHEMBL29014981 0.81 KCNH2 (0.61) KCNH2KMT2ACHEK2FYN
SCHEMBL30450304 0.81 KCNH2 (0.61) KCNH2KMT2ACHEK2FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116253687-A Diaryl pyrimidine compound and preparation method and application thereof 复旦大学 2023-06-13 CN disclosed