SCHEMBL30450993

SCHEMBL30450993

COC(=O)c1ccc2c(c1)C(=O)NC2

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 2/20 0.46
DYRK1B Q9Y463 2/20 0.46
NTRK2 Q16620 2/20 0.46
TYRO3 Q06418 1/20 0.46
FYN P06241 1/20 0.46
CASP3 P42574 1/20 0.46
JAK2 O60674 1/20 0.45
NTRK1 P04629 1/20 0.45
MET P08581 1/20 0.45
FGFR1 P11362 1/20 0.45
PRKACA P17612 1/20 0.45
KDR P35968 1/20 0.45
MAP2K2 P36507 1/20 0.45
FLT3 P36888 1/20 0.45
GSK3B P49841 1/20 0.45
MAP2K1 Q02750 1/20 0.45
MST1R Q04912 1/20 0.45
NTRK3 Q16288 1/20 0.45
CAMK1D Q8IU85 1/20 0.45
CA12 O43570 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19474641 1.00 CLK4 (0.46) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL31098601 0.88 SMYD3 (0.53) CLK4CASP3NTRK1PRKACAFLT3
SCHEMBL4611577 0.88 SMYD3 (0.53) CLK4CASP3NTRK1PRKACAFLT3
SCHEMBL14395236 0.85 PARP10 (0.56) CASP3PRKACACA12CA9CA1
SCHEMBL20446302 0.82 NPC1 (0.53) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL5879567 0.80 TDP2 (0.61) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL27491542 0.79 PRF1 (0.55) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL28367558 0.78 CLK4 (0.46) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL29873105 0.78 CLK4 (0.49) CLK4DYRK1BNTRK2TYRO3FYN
SCHEMBL24348699 0.77 CA12 (0.44) CLK4DYRK1BNTRK2TYRO3FYN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116261562-A PI 3K-alpha inhibitors and methods of use thereof 传达治疗有限公司 2023-06-13 CN disclosed