SCHEMBL30451193

SCHEMBL30451193

COc1ccc(CN2C(=O)c3cccc([N+](=O)[O-])c3C2=O)cc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 2/20 0.67
CA2 P00918 2/20 0.67
CA9 Q16790 2/20 0.67
CA12 O43570 1/20 0.67
KDM4E B2RXH2 2/20 0.60
CASP3 P42574 2/20 0.57
L3MBTL1 Q9Y468 2/20 0.55
TDP1 Q9NUW8 2/20 0.55
ALDH1A1 P00352 2/20 0.54
MAPT P10636 2/20 0.54
APEX1 P27695 1/20 0.54
MAOA P21397 1/20 0.53
CA4 P22748 1/20 0.53
POLB P06746 2/20 0.52
MEN1 O00255 2/20 0.52
KMT2A Q03164 2/20 0.52
HPGD P15428 1/20 0.52
MAPK1 P28482 1/20 0.52
ATM Q13315 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26712506 1.00 CA1 (0.67) CA1CA2CA9CA12KDM4E
SCHEMBL14348204 0.84 CA1 (0.73) CA1CA2CA9CA12KDM4E
SCHEMBL30305417 0.82 PARK7 (0.54) CA1CA2CA9CA12KDM4E
SCHEMBL5779243 0.81 CA1 (0.69) CA1CA2CA9CA12KDM4E
SCHEMBL16863040 0.81 CA1 (0.68) CA1CA2CA9CA12KDM4E
SCHEMBL23985223 0.81 KDM4E (0.76) KDM4ECASP3L3MBTL1ALDH1A1MAPT
SCHEMBL31667598 0.81 KDM4E (0.67) KDM4ECASP3L3MBTL1ALDH1A1MAPT
SCHEMBL18669037 0.81 CA9 (0.67) CA1CA2CA9CA12KDM4E
SCHEMBL20877391 0.80 KDM4E (0.65) KDM4ECASP3L3MBTL1ALDH1A1MAPT
SCHEMBL30428778 0.80 KDM4E (0.65) KDM4ECASP3L3MBTL1ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116261562-A PI 3K-alpha inhibitors and methods of use thereof 传达治疗有限公司 2023-06-13 CN disclosed