SCHEMBL30453293

SCHEMBL30453293

C#Cc1cnc(C(=O)NCC(=O)OC)c(OCOC)c1C

nearest known ligand 0.43

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGLN1 Q9GZT9 16/20 0.43
VEGFA P15692 4/20 0.43
FLT1 P17948 4/20 0.43
EGLN3 Q9H6Z9 3/20 0.43
KDM4E B2RXH2 1/20 0.34
GAA P10253 1/20 0.34
XDH P47989 1/20 0.34
GLA P06280 1/20 0.33
PKM P14618 1/20 0.33
STAMBP O95630 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26260159 0.92 SMN1; SMN2 (0.39) EGLN1VEGFAFLT1EGLN3KDM4E
SCHEMBL24257625 0.79 ALDH1A1 (0.39) EGLN1VEGFAFLT1EGLN3KDM4E
SCHEMBL26260156 0.78 SMN1; SMN2 (0.37) EGLN1VEGFAFLT1EGLN3KDM4E
SCHEMBL26260138 0.76 SMN1; SMN2 (0.43) EGLN1VEGFAFLT1EGLN3KDM4E
SCHEMBL26263986 0.75 EGLN1 (0.44) EGLN1VEGFAFLT1EGLN3GAA
SCHEMBL24257755 0.71 EGLN1 (0.55) EGLN1VEGFAFLT1EGLN3KDM4E
SCHEMBL26260298 0.70 EGLN1 (0.48) EGLN1VEGFAFLT1EGLN3KDM4E
SCHEMBL26260139 0.69 EGLN1 (0.42) EGLN1VEGFAFLT1EGLN3GAA
SCHEMBL30452393 0.68 SMN1; SMN2 (0.38) EGLN1VEGFAFLT1EGLN3GAA
SCHEMBL26260152 0.68 ALDH1A1 (0.41) EGLN1VEGFAFLT1EGLN3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4196466-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE Akebia Therapeutics Inc. (US) 2023-06-21 EP disclosed