SCHEMBL30453700

SCHEMBL30453700

Cc1c(-c2ccccn2)cnc(C(=O)O)c1O

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.43
KMT2A Q03164 1/20 0.43
KDM6B O15054 1/20 0.42
KDM4A O75164 1/20 0.42
KDM5C P41229 1/20 0.42
KDM4C Q9H3R0 1/20 0.42
KDM2A Q9Y2K7 1/20 0.42
KDM3A Q9Y4C1 1/20 0.42
PIN1 Q13526 1/20 0.39
BRD4 O60885 1/20 0.39
BRD2 P25440 1/20 0.39
BRD3 Q15059 1/20 0.39
BAZ2B Q9UIF8 1/20 0.39
BAZ2A Q9UIF9 1/20 0.39
P4HTM Q9NXG6 3/20 0.39
LMNA P02545 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
NAPRT Q6XQN6 1/20 0.39
ALDH1A1 P00352 3/20 0.38
MAOA P21397 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24257744 1.00 KDM4E (0.43) KDM4EKMT2AKDM6BKDM4AKDM5C
SCHEMBL24257547 0.82 EGLN2 (0.50)
SCHEMBL30546844 0.82 EGLN2 (0.50)
SCHEMBL25529048 0.77 KDM4E (0.46) KDM4EKMT2AKDM6BKDM4AKDM5C
SCHEMBL30546867 0.76 LMNA (0.50) KDM4ELMNAL3MBTL1ALDH1A1CYP1A2
SCHEMBL24257683 0.76 LMNA (0.50) KDM4ELMNAL3MBTL1ALDH1A1CYP1A2
SCHEMBL30453015 0.76 LMNA (0.50) KDM4ELMNAL3MBTL1ALDH1A1CYP1A2
SCHEMBL24257694 0.76 FYN (0.40) NAPRTERN1
SCHEMBL30546823 0.76 FYN (0.40) NAPRTERN1
SCHEMBL3387695 0.76 KDM4E (0.44) KDM4EKMT2AKDM6BKDM4AKDM5C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4196466-A1 PHD INHIBITOR COMPOUNDS, COMPOSITIONS, AND METHODS OF USE Akebia Therapeutics Inc. (US) 2023-06-21 EP disclosed