SCHEMBL30455909

SCHEMBL30455909

Nc1cc(-c2ccccn2)no1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.54
LMNA P02545 4/20 0.54
CCR1 P32246 3/20 0.54
CCR5 P51681 3/20 0.54
CCR8 P51685 3/20 0.54
BLM P54132 2/20 0.54
CYP1A2 P05177 1/20 0.54
POLB P06746 1/20 0.54
METAP1 P53582 1/20 0.54
HIF1A Q16665 1/20 0.54
DOHH Q9BU89 1/20 0.54
P4HTM Q9NXG6 1/20 0.54
ALDH1A1 P00352 4/20 0.49
MAPT P10636 4/20 0.49
TDO2 P48775 1/20 0.47
TP53 P04637 7/20 0.47
SMN1; SMN2 Q16637 6/20 0.47
NPC1 O15118 6/20 0.47
RAB9A P51151 5/20 0.47
PKM P14618 5/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2160804 1.00 KDM4E (0.54) KDM4ELMNACCR1CCR5CCR8
Benzamide SCHEMBL6318444 0.86 CHEK2 (0.49) KDM4ELMNACCR1CCR5CCR8
SCHEMBL4046101 0.77 KDM4E (0.54) KDM4ELMNACCR1CCR5CCR8
SCHEMBL3789967 0.77 KDM4E (0.54) KDM4ELMNACCR1CCR5CCR8
SCHEMBL2120922 0.77 NOTUM (0.62) KDM4ELMNACCR1CCR5CCR8
SCHEMBL224856 0.74 RAB9A (0.61) KDM4ELMNABLMCYP1A2ALDH1A1
Dipyridyl SCHEMBL29351528 0.73 KDM4E (1.00) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL3711450 0.73 KDM4E (1.00) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL29907716 0.73 KDM4E (1.00) KDM4ELMNACCR1CCR5CCR8
Dipyridyl SCHEMBL5922 0.73 KDM4E (1.00) KDM4ELMNACCR1CCR5CCR8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116438179-A Pyrazole derivatives as RET kinase inhibitors 伊莱利利公司 2023-07-14 CN disclosed