SCHEMBL30456364

SCHEMBL30456364

COC(=O)c1ccc2c(-c3nc(N[C@H]4CC[C@H](N)C4)ncc3C(F)(F)F)c[nH]c2c1Cl

nearest known ligand 0.51

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CCNE1 P24864 17/20 0.51
CDK2 P24941 17/20 0.51
CCNK O75909 17/20 0.51
CDK12 Q9NYV4 17/20 0.51
CCNT1 O60563 16/20 0.51
CDK9 P50750 16/20 0.51
CDK7 P50613 9/20 0.47
CCNH P51946 9/20 0.47
MNAT1 P51948 6/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25362625 1.00 CCNE1 (0.51) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL25362319 0.91 CCNK (0.51) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL30456473 0.91 CCNK (0.51) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL25364170 0.89 CCNK (0.56) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL31122407 0.89 CCNK (0.56) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL30456247 0.89 CCNK (0.56) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL30457188 0.89 CCNK (0.55) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL25360949 0.89 CCNK (0.55) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL25362356 0.88 CDK7 (0.48) CCNE1CDK2CCNKCDK12CCNT1
SCHEMBL30456173 0.88 CDK7 (0.48) CCNE1CDK2CCNKCDK12CCNT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250145632-A1 Pyrimidine Heterocyclic Compound, Preparation Method Thereof and use Thereof in Medicine INSILICO MEDICINE IP LIMITED (HK) 2025-05-08 US disclosed
EP-4455132-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE Insilico Medicine IP Limited (HK) 2024-10-30 EP disclosed
CN-118647607-A Pyrimidine heterocyclic compounds, process for preparing the same and pharmaceutical use thereof 英矽智能科技(上海)有限公司 2024-09-13 CN disclosed
WO-2023116761-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE 英矽智能科技知识产权有限公司 2023-06-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250145632-A1 Pyrimidine Heterocyclic Compound, Preparation Method Thereof and use Thereof in Medicine DPYD, TYMP, NUDT1 CCNE1 315/4885CDK2 73/4885CCNK 174/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.