SCHEMBL30456591

SCHEMBL30456591

CC(C)(C)OC(=O)N[C@H]1CC[C@H](Nc2ncc(C(F)(F)F)cn2)C1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HCRTR1 O43613 2/20 0.43
BTK Q06187 3/20 0.43
JAK1 P23458 5/20 0.42
KDM1A O60341 1/20 0.41
MAOB P27338 1/20 0.41
JAK2 O60674 2/20 0.41
CCRL2 O00421 1/20 0.40
MERTK Q12866 1/20 0.39
CKS1B P61024 1/20 0.39
SKP1 P63208 1/20 0.39
SKP2 Q13309 1/20 0.39
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
GAA P10253 1/20 0.38
SYK P43405 1/20 0.38
KMT2A Q03164 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
DRD2 P14416 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30995473 0.85 BTK (0.45) BTKJAK1KDM1AMAOBJAK2
SCHEMBL22241872 0.85 KDM1A (0.46) BTKJAK1KDM1AMAOBJAK2
SCHEMBL30842076 0.85 BTK (0.41) BTKJAK1KDM1AMAOBJAK2
SCHEMBL22406211 0.83 PCSK9 (0.50) BTKJAK1KDM1AMAOBJAK2
SCHEMBL22241734 0.83 PCSK9 (0.50) BTKJAK1KDM1AMAOBJAK2
SCHEMBL30842050 0.83 JAK1 (0.42) BTKJAK1KDM1AMAOBJAK2
SCHEMBL25360845 0.82 BTK (0.43) BTKJAK1KDM1AMAOBJAK2
SCHEMBL30456486 0.82 BTK (0.43) BTKJAK1KDM1AMAOBJAK2
SCHEMBL30827611 0.82 BTK (0.44) BTKJAK1KDM1AMAOBJAK2
SCHEMBL27252132 0.82 BTK (0.44) BTKJAK1KDM1AMAOBJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023116761-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE 英矽智能科技知识产权有限公司 2023-06-29 WO disclosed