SCHEMBL30456486

SCHEMBL30456486

CC(C)(C)OC(=O)N[C@H]1CC[C@H](Nc2ncc(C(F)(F)F)c(Cl)n2)C1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BTK Q06187 5/20 0.43
ULK1 O75385 2/20 0.40
JAK3 P52333 1/20 0.40
JAK1 P23458 3/20 0.38
LRRK2 Q5S007 2/20 0.38
JAK2 O60674 1/20 0.38
KDM1A O60341 1/20 0.38
MAOB P27338 1/20 0.38
MERTK Q12866 1/20 0.38
CKS1B P61024 1/20 0.37
SKP1 P63208 1/20 0.37
SKP2 Q13309 1/20 0.37
MAPK3 P27361 3/20 0.37
KMT2A Q03164 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25360845 1.00 BTK (0.43) BTKULK1JAK3JAK1LRRK2
SCHEMBL30456552 0.85 ULK1 (0.45) ULK1LRRK2MAPK3
SCHEMBL25362137 0.85 ULK1 (0.45) ULK1LRRK2MAPK3
SCHEMBL24087383 0.82 ULK1 (0.47) ULK1MAPK3EPHX2
SCHEMBL30456591 0.82 HCRTR1 (0.43) BTKJAK1JAK2KDM1AMAOB
SCHEMBL30842076 0.80 BTK (0.41) BTKJAK3JAK1JAK2KDM1A
SCHEMBL22901094 0.79 IDH1 (0.49) ULK1JAK1MAPK3L3MBTL1
SCHEMBL29821059 0.79 IDH1 (0.49) ULK1JAK1MAPK3L3MBTL1
SCHEMBL6460434 0.79 MCHR1 (0.48) ULK1JAK3MERTKCKS1BSKP1
SCHEMBL6460431 0.79 MCHR1 (0.48) ULK1JAK3MERTKCKS1BSKP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250145632-A1 Pyrimidine Heterocyclic Compound, Preparation Method Thereof and use Thereof in Medicine INSILICO MEDICINE IP LIMITED (HK) 2025-05-08 US disclosed
EP-4455132-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE Insilico Medicine IP Limited (HK) 2024-10-30 EP disclosed
WO-2023116761-A1 PYRIMIDINE HETEROCYCLIC COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF IN MEDICINE 英矽智能科技知识产权有限公司 2023-06-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250145632-A1 Pyrimidine Heterocyclic Compound, Preparation Method Thereof and use Thereof in Medicine DPYD, TYMP, NUDT1 BTK 162/4885ULK1 2923/4885JAK3 75/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.