SCHEMBL30456780

SCHEMBL30456780

C[Si](C)(C)CCOCn1cc(Br)c2c(Cl)ccnc21

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 5/20 0.40
MPO P05164 1/20 0.31
TPO P07202 1/20 0.31
KCNH2 Q12809 1/20 0.31
NPC1 O15118 1/20 0.30
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25239242 1.00 DGAT1 (0.40) DGAT1MPOTPOKCNH2NPC1
SCHEMBL21678682 1.00 DGAT1 (0.40) DGAT1MPOTPOKCNH2NPC1
SCHEMBL30457445 0.88 DGAT1 (0.42) DGAT1NPC1
SCHEMBL14158745 0.88 DGAT1 (0.42) DGAT1NPC1
SCHEMBL29854683 0.86 DGAT1 (0.38) DGAT1MAPT
SCHEMBL2693867 0.86 DGAT1 (0.38) DGAT1MAPT
SCHEMBL2238008 0.85 DGAT1 (0.35) DGAT1MAPT
SCHEMBL30295772 0.85 DGAT1 (0.35) DGAT1MAPT
SCHEMBL21632538 0.85 DGAT1 (0.45) DGAT1NPC1
SCHEMBL2696013 0.84 DGAT1 (0.35) DGAT1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-119080779-A Pyrrolopyrimidine ITK inhibitors 阿克拉瑞斯治疗股份有限公司 2024-12-06 CN disclosed
CN-112823005-B Pyrrolopyrimidine ITK inhibitors 阿克拉瑞斯治疗股份有限公司 2024-08-20 CN disclosed
WO-2023110843-A1 HETEROBICYCLIC DERIVATIVES AS ITK INHIBITORS ALMIRALL, S.A. (ES) 2023-06-22 WO disclosed