SCHEMBL30459722

SCHEMBL30459722

CCOc1ccc2c(cnn2-c2ccnc(Nc3cc([N+](=O)[O-])c(F)cc3OC)n2)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.54
EGFR P00533 5/20 0.41
MAPK8 P45983 2/20 0.36
MAPK10 P53779 2/20 0.36
NR3C1 P04150 2/20 0.35
MEN1 O00255 2/20 0.35
HPGD P15428 2/20 0.35
KMT2A Q03164 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2C9 P11712 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
CCNT1 O60563 2/20 0.35
CDK1 P06493 2/20 0.35
CCNB1 P14635 2/20 0.35
CDK9 P50750 2/20 0.35
CDK7 P50613 1/20 0.35
CCNH P51946 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
MAPT P10636 3/20 0.35
MAPK9 P45984 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683364 1.00 KDR (0.54) KDREGFRMAPK8MAPK10NR3C1
SCHEMBL17683144 0.94 KDR (0.57) KDREGFRMAPK8MAPK10MEN1
SCHEMBL30459859 0.94 KDR (0.57) KDREGFRMAPK8MAPK10MEN1
SCHEMBL30460247 0.87 KDR (0.54) KDREGFRMAPK8MAPK10MEN1
SCHEMBL17683109 0.87 KDR (0.54) KDREGFRMAPK8MAPK10MEN1
SCHEMBL17683366 0.86 EGFR (0.51) KDREGFR
SCHEMBL19254873 0.86 KDR (0.54) KDREGFRMAPK8MAPK10CCNT1
SCHEMBL17683359 0.86 KDR (0.54) KDREGFRMAPK8MAPK10CCNT1
SCHEMBL17683292 0.82 MAPK8 (0.53) KDREGFRMAPK8MAPK10CCNT1
SCHEMBL17683143 0.81 EGFR (0.53) KDREGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
CN-111187221-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-26 CN disclosed
CN-111171000-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed
CN-111170999-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed