SCHEMBL30459859

SCHEMBL30459859

COc1ccc2c(cnn2-c2ccnc(Nc3cc([N+](=O)[O-])c(F)cc3OC)n2)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 2/20 0.57
EGFR P00533 2/20 0.41
CCNT1 O60563 2/20 0.37
CDK1 P06493 2/20 0.37
CCNB1 P14635 2/20 0.37
CDK9 P50750 2/20 0.37
CDK7 P50613 1/20 0.37
CCNH P51946 1/20 0.37
MKNK2 Q9HBH9 4/20 0.37
MEN1 O00255 4/20 0.36
KMT2A Q03164 4/20 0.36
MKNK1 Q9BUB5 2/20 0.36
MAPT P10636 4/20 0.36
GAA P10253 1/20 0.36
MAPK1 P28482 1/20 0.36
CCNA2 P20248 1/20 0.36
CDK2 P24941 1/20 0.36
TTK P33981 1/20 0.36
MAPK8 P45983 1/20 0.36
MAPK9 P45984 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683144 1.00 KDR (0.57) KDREGFRCCNT1CDK1CCNB1
SCHEMBL30459722 0.94 KDR (0.54) KDREGFRCCNT1CDK1CCNB1
SCHEMBL17683364 0.94 KDR (0.54) KDREGFRCCNT1CDK1CCNB1
SCHEMBL17683109 0.90 KDR (0.54) KDREGFRCCNT1CDK1CCNB1
SCHEMBL30460247 0.90 KDR (0.54) KDREGFRCCNT1CDK1CCNB1
SCHEMBL19254873 0.89 KDR (0.54) KDREGFRCCNT1CDK1CCNB1
SCHEMBL17683359 0.89 KDR (0.54) KDREGFRCCNT1CDK1CCNB1
SCHEMBL17683143 0.85 EGFR (0.53) KDREGFR
SCHEMBL17683292 0.85 MAPK8 (0.53) KDREGFRCCNT1CDK1CCNB1
SCHEMBL17683302 0.84 KDR (0.41) KDREGFRMKNK2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
CN-111187221-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-26 CN disclosed
CN-111171000-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed
CN-111170999-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed