SCHEMBL30459758

SCHEMBL30459758

COc1cc2[nH]nc(C)c2cc1OC

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.50
ADORA2B P29275 1/20 0.50
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 3/20 0.46
HPGD P15428 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
PDE3A Q14432 3/20 0.42
PDE10A Q9Y233 1/20 0.42
GRIN2D O15399 1/20 0.41
GRIN3B O60391 1/20 0.41
GRIN1 Q05586 1/20 0.41
GRIN2A Q12879 1/20 0.41
GRIN2B Q13224 1/20 0.41
GRIN2C Q14957 1/20 0.41
GRIN3A Q8TCU5 1/20 0.41
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
AURKA O14965 1/20 0.39
PDE3B Q13370 2/20 0.39
MAPT P10636 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683153 1.00 ADORA2A (0.50) ADORA2AADORA2BKDM4EALDH1A1HPGD
SCHEMBL11708958 0.80 KDM4E (0.46) KDM4EALDH1A1HPGDSMN1; SMN2GRIN2D
Hydrochloric Acid SCHEMBL11708649 0.78 KDM4E (0.45) KDM4EALDH1A1HPGDSMN1; SMN2GRIN2D
SCHEMBL16867222 0.78 ADORA2A (0.67) ADORA2AADORA2BAURKACDK4CCNA2
SCHEMBL11546262 0.77 PDE4A (0.49) KDM4EALDH1A1HPGDSMN1; SMN2PDE3A
SCHEMBL14297421 0.76 ADORA2A (0.59) ADORA2AADORA2BKDM4EALDH1A1HPGD
SCHEMBL27927364 0.76 ALDH1A1 (0.42) KDM4EALDH1A1HPGDSMN1; SMN2PDE3A
SCHEMBL11750245 0.76 ALDH1A1 (0.42) KDM4EALDH1A1HPGDSMN1; SMN2PDE3A
SCHEMBL15540970 0.74 NTRK1 (0.49) KDM4EALDH1A1HPGDSMN1; SMN2PDE3A
SCHEMBL28141790 0.74 ALDH1A1 (0.41) KDM4EALDH1A1HPGDSMN1; SMN2PDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
CN-111187221-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-26 CN disclosed
CN-111171000-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed
CN-111170999-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed