SCHEMBL30459760

SCHEMBL30459760

COc1ccc2c(cnn2-c2ccnc(S(C)(=O)=O)n2)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP11B1 P15538 2/20 0.43
CYP11B2 P19099 2/20 0.43
KDR P35968 2/20 0.41
ROCK1 Q13464 2/20 0.41
MAPT P10636 1/20 0.38
PIM3 Q86V86 1/20 0.37
CCNT1 O60563 2/20 0.36
CDK1 P06493 2/20 0.36
CCNB1 P14635 2/20 0.36
CDK9 P50750 2/20 0.36
NR3C1 P04150 2/20 0.36
CDK7 P50613 1/20 0.36
CCNH P51946 1/20 0.36
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
NPC1 O15118 2/20 0.36
RAB9A P51151 2/20 0.36
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
MEN1 O00255 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683145 1.00 CYP11B1 (0.43) CYP11B1CYP11B2KDRROCK1MAPT
SCHEMBL30459679 0.88 NR3C1 (0.42) CYP11B1CYP11B2KDRMAPTCCNT1
SCHEMBL17683288 0.88 NR3C1 (0.42) CYP11B1CYP11B2KDRMAPTCCNT1
SCHEMBL5090337 0.84 CYP11B1 (0.40) CYP11B1CYP11B2KDRROCK1CCNT1
SCHEMBL3823223 0.80 CDK1 (0.53) CYP11B1CYP11B2CCNT1CDK1CCNB1
SCHEMBL17683115 0.79 LRRK2 (0.40) KDRPIM3CCNT1CDK1CCNB1
SCHEMBL17683138 0.78 ROCK1 (0.45) CYP11B1CYP11B2KDRROCK1MAPT
SCHEMBL30459759 0.78 ROCK1 (0.45) CYP11B1CYP11B2KDRROCK1MAPT
SCHEMBL17683301 0.78 DYRK1A (0.45) ROCK1PIM3CCNT1CDK1CCNB1
SCHEMBL5102689 0.77 IRAK4 (0.44) CCNT1CDK1CCNB1CDK9CDK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
CN-111187221-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-26 CN disclosed
CN-111171000-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed
CN-111170999-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed