SCHEMBL30459855

SCHEMBL30459855

COc1cc(N2CC3(COC3)C2)c(C=CC(N)=O)cc1Nc1nccc(-c2cn(C)c3ccccc23)n1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.57
MKNK1 Q9BUB5 1/20 0.53
MKNK2 Q9HBH9 1/20 0.53
MLNR O43193 1/20 0.50
KDM1A O60341 1/20 0.50
ABCB11 O95342 1/20 0.50
ERBB2 P04626 1/20 0.50
INSR P06213 1/20 0.50
CHRM2 P08172 1/20 0.50
HTR1A P08908 1/20 0.50
ADORA3 P0DMS8 1/20 0.50
DRD2 P14416 1/20 0.50
NQO2 P16083 1/20 0.50
ADRA2C P18825 1/20 0.50
DRD1 P21728 1/20 0.50
ERBB3 P21860 1/20 0.50
SLC6A2 P23975 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
ADORA2A P29274 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17683051 0.84 EGFR (0.80) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL30539153 0.82 EGFR (0.61) EGFRMKNK1MKNK2KCNH2IGF1R
SCHEMBL30460261 0.81 EGFR (0.61) EGFRMKNK1MKNK2MLNRKDM1A
SCHEMBL16877321 0.80 EGFR (0.73) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL17683067 0.78 EGFR (0.83) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL20854998 0.78 EGFR (0.74) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL19540857 0.75 EGFR (0.64) EGFRMKNK1MKNK2MLNRKDM1A
SCHEMBL19540924 0.75 EGFR (0.72) EGFRMKNK1MKNK2MLNRKDM1A
SCHEMBL19254808 0.74 EGFR (0.87) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL18870128 0.74 MKNK2 (0.75) EGFRMKNK1MKNK2MLNRKDM1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117402143-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2024-01-16 CN disclosed
CN-117069700-A EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-11-17 CN disclosed
CN-111187221-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-26 CN disclosed
CN-111171000-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-09-01 CN disclosed
CN-111170999-B EGFR inhibitor and preparation and application thereof 上海翰森生物医药科技有限公司 2023-06-30 CN disclosed