SCHEMBL30459975

SCHEMBL30459975

COC(=O)c1ccc2c(c1)C(C)(C)C(=O)N2

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 6/20 0.51
PDE3B Q13370 2/20 0.48
PDE3A Q14432 2/20 0.48
PDK2 Q15119 1/20 0.46
PDK4 Q16654 1/20 0.46
IP6K1 Q92551 1/20 0.46
LMNA P02545 2/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPT P10636 2/20 0.45
CA12 O43570 1/20 0.45
CA1 P00915 1/20 0.45
CA2 P00918 1/20 0.45
CA7 P43166 1/20 0.45
XDH P47989 1/20 0.45
CA9 Q16790 1/20 0.45
CA14 Q9ULX7 1/20 0.45
ALOX5 P09917 1/20 0.43
KIF11 P52732 1/20 0.43
MEN1 O00255 1/20 0.42
FGB P02675 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29041890 1.00 PGR (0.51) PGRPDE3BPDE3APDK2PDK4
SCHEMBL16321516 0.88 MAPK14 (0.53) PGRPDK2PDK4LMNAALDH1A1
SCHEMBL29825095 0.88 MAPK14 (0.53) PGRPDK2PDK4LMNAALDH1A1
SCHEMBL4904403 0.83 IP6K1 (0.45) PDK2IP6K1LMNAALDH1A1MAPT
SCHEMBL1874397 0.82 PGR (0.55) PGRPDE3BPDE3APDK2PDK4
SCHEMBL25156270 0.80 MAPK14 (0.43) PGRPDE3BPDE3APDK2PDK4
SCHEMBL12548325 0.79 IP6K1 (0.57) PGRPDE3BPDE3AIP6K1LMNA
SCHEMBL7379550 0.78 PGR (0.51) PGRPDE3BPDE3APDK2PDK4
SCHEMBL31117105 0.78 PGR (0.51) PGRPDE3BPDE3APDK2PDK4
SCHEMBL22711811 0.77 IP6K1 (0.56) IP6K1LMNAALDH1A1MAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116457346-A Preparation of indolone derivatives as novel diacylglycerol O-acyltransferase 2 inhibitors 默沙东有限责任公司 2023-07-18 CN disclosed