Gsk-300014A

Gsk-300014A

SCHEMBL30467447

CS(=O)(=O)CCNCc1cc(-c2cc3c(Nc4ccc(OCc5cccc(F)c5)c(Cl)c4)ncnc3s2)cs1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 20/20 1.00
ERBB2 P04626 18/20 1.00
MEN1 O00255 3/20 0.66
KMT2A Q03164 3/20 0.66
MAPK1 P28482 2/20 0.66
CYP3A4 P08684 2/20 0.65
KDM4E B2RXH2 1/20 0.65
ALDH1A1 P00352 1/20 0.65
MAPT P10636 1/20 0.65
ALOX15 P16050 1/20 0.65
HSD17B10 Q99714 1/20 0.65
PIK3C2B O00750 1/20 0.64
MAP2K7 O14733 1/20 0.64
RIPK2 O43353 1/20 0.64
PIK3C2G O75747 1/20 0.64
STK10 O94804 1/20 0.64
ABCB11 O95342 1/20 0.64
ABL1 P00519 1/20 0.64
INSR P06213 1/20 0.64
RET P07949 1/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6496570 0.80 EGFR (0.69) EGFRERBB2MEN1KMT2AMAPK1
SCHEMBL5069008 0.80 EGFR (0.67) EGFRERBB2MEN1KMT2AMAPK1
SCHEMBL114539 0.80 EGFR (1.00) EGFRERBB2MEN1KMT2AMAPK1
SCHEMBL5064133 0.79 EGFR (0.66) EGFRERBB2MEN1KMT2AMAPK1
Hydrochloric Acid SCHEMBL30362906 0.79 EGFR (1.00) EGFRERBB2MEN1KMT2AMAPK1
Hydrochloric Acid SCHEMBL29556740 0.79 EGFR (1.00) EGFRERBB2MEN1KMT2AMAPK1
Hydrochloric Acid SCHEMBL9988095 0.79 EGFR (1.00) EGFRERBB2MEN1KMT2AMAPK1
SCHEMBL2099770 0.78 EGFR (0.83) EGFRERBB2MEN1KMT2AMAPK1
SCHEMBL14264605 0.78 EGFR (0.90) EGFRERBB2MEN1KMT2ACYP3A4
Lapatinib SCHEMBL29464189 0.78 EGFR (1.00) EGFRERBB2MEN1KMT2ACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230190748-A1 COMPOSITIONS FOR TREATMENT OF AGED DISEASES GERO PTE LTD (SG) 2023-06-22 US claimed
US-20230190748-A1 COMPOSITIONS FOR TREATMENT OF AGED DISEASES GERO PTE LTD (SG) 2023-06-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230190748-A1 COMPOSITIONS FOR TREATMENT OF AGED DISEASES AGER, CKMT1A; CKMT1B, GLA EGFR 1153/4885ERBB2 1599/4885MEN1 3801/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.