SCHEMBL30468458

SCHEMBL30468458

CC1Cc2ccccc2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.45

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.45
NR1H2 P55055 1/20 0.45
PRMT5 O14744 4/20 0.45
WDR77 Q9BQA1 4/20 0.45
DRD2 P14416 4/20 0.43
GPR119 Q8TDV5 1/20 0.43
ESR2 Q92731 1/20 0.43
UCHL1 P09936 1/20 0.43
ALDH1A1 P00352 1/20 0.42
NAMPT P43490 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
NOTUM Q6P988 1/20 0.41
KDM1A O60341 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29376321 0.87 NAMPT (0.48) MAPK1PRMT5WDR77DRD2NAMPT
SCHEMBL12013723 0.87 NAMPT (0.48) MAPK1PRMT5WDR77DRD2NAMPT
SCHEMBL14138611 0.87 NAMPT (0.48) MAPK1PRMT5WDR77DRD2NAMPT
SCHEMBL29051832 0.85 ESR2 (0.63) NR1H2DRD2ESR2
SCHEMBL29052424 0.84 NR1H2 (0.64) NR1H2ESR2KDM1A
SCHEMBL30468516 0.83 ESR2 (0.47) NR1H2DRD2ESR2ALDH1A1NOTUM
SCHEMBL1791198 0.83 UCHL1 (0.48) MAPK1NR1H2PRMT5WDR77GPR119
SCHEMBL19389912 0.83 DRD1 (0.53) MAPK1NR1H2PRMT5WDR77DRD2
SCHEMBL29705902 0.83 DRD1 (0.53) MAPK1NR1H2PRMT5WDR77DRD2
SCHEMBL30429426 0.80 PRMT5 (0.43) MAPK1NR1H2PRMT5WDR77DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116332910-A 2-aminopyrimidine derivatives as kinase inhibitors, preparation and use thereof 江苏威凯尔医药科技有限公司 2023-06-27 CN disclosed