SCHEMBL30475035

SCHEMBL30475035

COC(=O)c1nc(C(F)(F)F)c(Br)cc1NC(C)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.40
CYP1A2 P05177 3/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
NPSR1 Q6W5P4 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
ATM Q13315 1/20 0.39
PTPN2 P17706 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
SOS1 Q07889 1/20 0.36
DYRK1A Q13627 2/20 0.35
MAPT P10636 2/20 0.35
NPC1 O15118 1/20 0.34
PKM P14618 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25305491 1.00 NOTUM (0.40) NOTUMCYP1A2CYP2C9CYP2C19NPSR1
SCHEMBL25307557 0.86 CA1 (0.35) CYP1A2CYP2C9CYP2C19NPSR1CYP3A4
SCHEMBL30475042 0.82 NOTUM (0.34) NOTUMNPSR1PTPN2ALDH1A1SOS1
SCHEMBL25299508 0.82 NOTUM (0.34) NOTUMNPSR1PTPN2ALDH1A1SOS1
SCHEMBL31214172 0.80 NOTUM (0.43) NOTUMNPSR1PTPN2ALDH1A1SOS1
SCHEMBL25304722 0.80 ALDH1A1 (0.40) CYP1A2NPSR1ALDH1A1CA1CA2
SCHEMBL30475022 0.80 ALDH1A1 (0.40) CYP1A2NPSR1ALDH1A1CA1CA2
SCHEMBL25263446 0.79 CFTR (0.48) NOTUMNPSR1PTPN2SOS1CFTR
SCHEMBL30664857 0.79 CFTR (0.48) NOTUMNPSR1PTPN2SOS1CFTR
SCHEMBL25305667 0.78 SOS1 (0.45) NOTUMCYP1A2PTPN2ALDH1A1SOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023225252-A1 COMPOSITIONS AND METHODS FOR INHIBITION OF RAS THERAS, INC. (US) 2023-11-23 WO disclosed
WO-2023133183-A1 KRAS INHIBITORS THERAS, INC. (US) 2023-07-13 WO disclosed