SCHEMBL30484385

SCHEMBL30484385

O=c1[nH]n(-c2ccccn2)c2ncncc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.60
MAPK1 P28482 1/20 0.60
LDHA P00338 1/20 0.48
CHEK1 O14757 1/20 0.44
AURKA O14965 1/20 0.44
DAPK3 O43293 1/20 0.44
JAK2 O60674 1/20 0.44
PRKD3 O94806 1/20 0.44
MAP4K4 O95819 1/20 0.44
PAK4 O96013 1/20 0.44
ABL1 P00519 1/20 0.44
NTRK1 P04629 1/20 0.44
FYN P06241 1/20 0.44
CSF1R P07333 1/20 0.44
RET P07949 1/20 0.44
IGF1R P08069 1/20 0.44
MET P08581 1/20 0.44
PDGFRB P09619 1/20 0.44
PIM1 P11309 1/20 0.44
FGFR1 P11362 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30613317 0.80 HPGD (0.39) GAAMAPK1LDHANTRK1HPGD
SCHEMBL30305668 0.76 GAA (0.55) GAAMAPK1LDHACHEK1AURKA
SCHEMBL30378078 0.76 WEE1 (0.54)
SCHEMBL21296397 0.76 WEE1 (0.54)
SCHEMBL11411739 0.75 GAA (1.00) GAAMAPK1LDHACHEK1AURKA
Hydrochloric Acid SCHEMBL30561520 0.75 WEE1 (0.53)
SCHEMBL30613291 0.74 GAA (0.52) GAAMAPK1LDHACHEK1AURKA
SCHEMBL23038644 0.74 WEE1 (0.42) GAAMAPK1LDHANTRK1CLK4
SCHEMBL4707558 0.68 KDM4E (0.39) MAPK1CLK4CYP1A2CYP2C19CYP2C9
SCHEMBL30057955 0.68 KDM4E (0.39) MAPK1CLK4CYP1A2CYP2C19CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117720541-A Substituted 1, 2-dihydro-3H-pyrazolo [3,4-d ] pyrimidin-3-ones 里科瑞尔姆IP控股有限责任公司 2024-03-19 CN disclosed
CN-116947890-A Tricyclic compound of WEE1 inhibitor, and preparation method and application thereof 星希尔生物科技(上海)有限公司 2023-10-27 CN disclosed
CN-111902413-B Substituted 1, 2-dihydro-3H-pyrazolo [3,4-d ] pyrimidin-3-ones 里科瑞尔姆IP控股有限责任公司 2023-10-17 CN disclosed
CN-112142748-B Pyrazolopyrimidine compound, and preparation method and application thereof 上海医药集团股份有限公司 2023-07-04 CN disclosed