SCHEMBL30487302

SCHEMBL30487302

COc1ccc(Cn2ncc3ccc(Br)nc32)cc1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 9/20 0.48
PDE1B Q01064 4/20 0.46
PDE1A P54750 3/20 0.46
PDE1C Q14123 3/20 0.46
MCHR1 Q99705 1/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
MAPT P10636 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
HPGD P15428 1/20 0.42
ALOX15 P16050 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
HSD17B10 Q99714 1/20 0.42
BRD4 O60885 1/20 0.42
MET P08581 1/20 0.41
CNR2 P34972 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29071647 1.00 NPBWR1 (0.48) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL30731296 0.84 NPBWR1 (0.52) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL15545682 0.84 NPBWR1 (0.52) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL21796911 0.83 NPBWR1 (0.48) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL21796474 0.79 NPBWR1 (0.44) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL22553999 0.79 CNR2 (0.55) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL30731305 0.79 CNR2 (0.55) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL2961568 0.78 PDE1B (0.52) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL17395029 0.78 NPBWR1 (0.48) NPBWR1PDE1BPDE1APDE1CMCHR1
SCHEMBL5091051 0.77 BRD4 (0.53) NPBWR1PDE1BPDE1APDE1CMCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116535401-A Novel PARP1 inhibitors and uses thereof 南京圣和药业股份有限公司 2023-08-04 CN disclosed