SCHEMBL30489596

SCHEMBL30489596

CC(=O)SCC(C)(C)NC(=O)OC(C)(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.36
CA1 P00915 2/20 0.35
CA2 P00918 2/20 0.35
CA7 P43166 2/20 0.35
MEN1 O00255 1/20 0.34
GAA P10253 1/20 0.34
KMT2A Q03164 1/20 0.34
CA12 O43570 2/20 0.33
CA14 Q9ULX7 2/20 0.33
APLNR P35414 1/20 0.33
IDO1 P14902 1/20 0.32
CTSK P43235 2/20 0.32
MAOA P21397 1/20 0.32
MAOB P27338 1/20 0.32
CYP2D6 P10635 1/20 0.32
LATS1 O95835 1/20 0.32
DGAT1 O75907 1/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4754596 0.81 TDP1 (0.38) TDP1CA1CA2CA7MEN1
SCHEMBL18340829 0.81 MEN1 (0.35) TDP1CA1CA2CA7MEN1
SCHEMBL14280309 0.78 TDP1 (0.38) TDP1CA1CA2CA7MEN1
SCHEMBL15426303 0.78 CYP2C19 (0.32) CYP2C19
SCHEMBL14845755 0.76 TDP1 (0.33) TDP1CA1CA2MEN1GAA
SCHEMBL21261831 0.76 TDP1 (0.42) TDP1CA1CA2CA7MEN1
SCHEMBL2870572 0.75 CYP1A2 (0.32) CA2CA12CA14CYP1A2CYP2C9
SCHEMBL1233866 0.75 TDP1 (0.39) TDP1CA1CA2CA7MEN1
SCHEMBL57379 0.74 TDP1 (0.46) TDP1CA1CA2CA7MEN1
SCHEMBL4616898 0.74 CA1 (0.42) TDP1CA1CA2CA7MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3313828-B1 METALLO-BETA-LACTAMASE INHIBITORS MERCK SHARP & DOHME LLC (US) 2023-07-12 EP disclosed