SCHEMBL3049527

SCHEMBL3049527

CN1CCN(C(=O)C(Cc2ccccc2)NC(=O)C(CCCCNC(=O)OC(C)(C)C)NC(=O)OCC2c3ccccc3-c3ccccc32)CC1

nearest known ligand 0.61

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TLR2 O60603 1/20 0.48
TLR1 Q15399 1/20 0.48
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
MDM2 Q00987 1/20 0.45
HRH2 P25021 1/20 0.45
HRH1 P35367 1/20 0.45
PAX8 Q06710 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
KMT2A Q03164 3/20 0.44
TGM2 P21980 2/20 0.43
PTPN1 P18031 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29431191 0.88 MDM2 (0.51) TLR2TLR1MDM2PAX8TDP1
SCHEMBL13702142 0.88 TLR2 (0.53) TLR2TLR1ITGB3ITGA2BMDM2
SCHEMBL8259207 0.87 PAX8 (0.50) TLR2TLR1MDM2PAX8TDP1
SCHEMBL12340097 0.86 KMT2A (0.48) TLR2TLR1MDM2PAX8TDP1
SCHEMBL30193403 0.86 MDM2 (0.52) TLR2TLR1MDM2PAX8TDP1
SCHEMBL1755616 0.86 PAX8 (0.55) TLR2TLR1MDM2PAX8TDP1
SCHEMBL16870156 0.86 MDM2 (0.52) TLR2TLR1MDM2PAX8TDP1
SCHEMBL18421240 0.86 MDM2 (0.52) TLR2TLR1MDM2PAX8TDP1
SCHEMBL30193389 0.86 MDM2 (0.52) TLR2TLR1MDM2PAX8TDP1
SCHEMBL16870002 0.86 MDM2 (0.52) TLR2TLR1MDM2PAX8TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7745413-B2 Collection of traceable compounds and uses thereof CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2010-06-29 US disclosed
US-20080176763-A1 Collection of Traceable Compounds and Uses Thereof CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (FR) 2008-07-24 US disclosed