SCHEMBL30495481

SCHEMBL30495481

CCCn1c(=O)[nH]c(N)c(NC(=O)c2cnn(Cc3cccc(C(F)(F)F)c3)c2)c1=O

nearest known ligand 0.58

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 19/20 0.58
ADORA2A P29274 14/20 0.58
ADORA3 P0DMS8 11/20 0.58
ADORA1 P30542 13/20 0.52
PLK4 O00444 1/20 0.50
CDK2 P24941 1/20 0.50
IRAK1 P51617 1/20 0.50
RPS6KA3 P51812 1/20 0.50
PLK3 Q9H4B4 1/20 0.50
CSNK1G3 Q9Y6M4 1/20 0.50
SCD5 Q86SK9 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL796431 1.00 ADORA2B (0.58) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1546106 0.90 ADORA2B (0.58) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1546641 0.89 ADORA2B (0.56) ADORA2BADORA2AADORA3ADORA1SCD5
SCHEMBL8979404 0.88 ADORA2B (0.49) ADORA2BADORA2AADORA3ADORA1
SCHEMBL1546614 0.87 ADORA2B (0.59) ADORA2BADORA2AADORA3ADORA1SCD5
SCHEMBL5541331 0.87 ADORA2B (0.45) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1723697 0.87 ADORA2B (0.52) ADORA2BADORA2AADORA3ADORA1RPS6KA3
SCHEMBL1546107 0.87 ADORA2B (0.54) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL244147 0.86 ADORA2B (0.55) ADORA2BADORA2AADORA3ADORA1PLK4
SCHEMBL1546781 0.85 KLKB1 (0.52) ADORA2BADORA2AADORA3ADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111770926-B Tricyclic compounds, compositions and pharmaceutical uses thereof 因佩蒂斯生物科学有限公司 2023-07-21 CN disclosed