SCHEMBL30507464

SCHEMBL30507464

COc1ccc(-c2ccnc(N)n2)c(OC)c1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.60
DYRK1A Q13627 2/20 0.60
MAP3K14 Q99558 1/20 0.60
CHRNA7 P36544 1/20 0.53
CYP1A1 P04798 1/20 0.52
CYP1B1 Q16678 1/20 0.52
CCNT1 O60563 3/20 0.52
CDK2 P24941 3/20 0.52
CDK9 P50750 3/20 0.52
CDK5 Q00535 2/20 0.52
CDK5R1 Q15078 2/20 0.52
CCNA2 P20248 2/20 0.52
CCNA1 P78396 1/20 0.52
TLR9 Q9NR96 2/20 0.50
CRHR1 P34998 1/20 0.50
HTR1A P08908 1/20 0.50
HTR7 P34969 1/20 0.50
HTR2B P41595 1/20 0.50
HTR5A P47898 1/20 0.50
TLR7 Q9NYK1 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28512792 1.00 GSK3B (0.60) GSK3BDYRK1AMAP3K14CHRNA7CYP1A1
SCHEMBL5471286 0.88 GSK3B (0.60) GSK3BDYRK1AMAP3K14CCNT1CDK2
SCHEMBL3658285 0.86 CCNT1 (0.53) GSK3BDYRK1AMAP3K14CCNT1CDK2
SCHEMBL28497712 0.85 CDK2 (0.52) GSK3BDYRK1AMAP3K14CCNT1CDK2
SCHEMBL30507501 0.85 CDK2 (0.52) GSK3BDYRK1AMAP3K14CCNT1CDK2
SCHEMBL30451078 0.84 CYP1A1 (0.55) CYP1A1CYP1B1TLR9CRHR1TLR7
SCHEMBL12306207 0.84 HSP90AA1 (0.59) DYRK1ACHRNA7CYP1A1CYP1B1TLR9
SCHEMBL15939816 0.84 CHRNA7 (0.55) GSK3BDYRK1AMAP3K14CHRNA7CCNT1
SCHEMBL30507254 0.84 CHRNA7 (0.55) GSK3BDYRK1AMAP3K14CHRNA7CCNT1
SCHEMBL444455 0.82 CYP1A1 (0.52) CYP1A1CYP1B1CCNT1CDK9TLR9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112010844-B Preparation method and application of N- (pyrimidine-2-yl) coumarin-7-amine derivative as protein kinase inhibitor 中国药科大学 2023-07-25 CN disclosed