SCHEMBL3658285

SCHEMBL3658285

COc1cc(N)ccc1-c1ccnc(N)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 6/20 0.53
CDK9 P50750 6/20 0.53
CDK5 Q00535 5/20 0.53
CDK5R1 Q15078 5/20 0.53
CCNA2 P20248 5/20 0.53
CDK2 P24941 5/20 0.53
CCNA1 P78396 3/20 0.53
GSK3B P49841 2/20 0.51
DYRK1A Q13627 2/20 0.51
HTR1A P08908 1/20 0.51
HTR7 P34969 1/20 0.51
HTR2B P41595 1/20 0.51
HTR5A P47898 1/20 0.51
NFATC1 O95644 1/20 0.51
KDM4E B2RXH2 2/20 0.49
ALDH1A1 P00352 1/20 0.49
RAB9A P51151 1/20 0.49
MAP3K14 Q99558 1/20 0.48
HSP90AA1 P07900 3/20 0.47
HSP90AB1 P08238 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30507501 0.86 CDK2 (0.52) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL28512792 0.86 GSK3B (0.60) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL30507464 0.86 GSK3B (0.60) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL28497712 0.86 CDK2 (0.52) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL31011620 0.85 HSP90AA1 (0.45) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL31011609 0.85 HSP90AA1 (0.45) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL30507254 0.85 CHRNA7 (0.55) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL15939816 0.85 CHRNA7 (0.55) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL30507329 0.81 HSP90AA1 (0.60) CCNT1CDK9CDK5CDK5R1CCNA2
SCHEMBL3362587 0.81 HSP90AA1 (0.60) CCNT1CDK9CDK5CDK5R1CCNA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2234618-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS The Scripps Research Institute (US) 2010-10-06 EP disclosed
WO-2009079008-A1 BENZOPYRANS AND ANALOGS AS RHO KINASE INHIBITORS FENG YANGBO (US) 2009-06-25 WO disclosed