SCHEMBL30514765

SCHEMBL30514765

CC(=O)Nc1cc(-c2cc(OC(C)(C)C)nc(-c3cccnc3C(F)(F)F)c2)ccn1

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TGFBR1 P36897 3/20 0.43
AAK1 Q2M2I8 7/20 0.43
CYP3A4 P08684 6/20 0.43
PIK3C3 Q8NEB9 7/20 0.41
TGFBR2 P37173 2/20 0.40
ADORA3 P0DMS8 2/20 0.39
ADORA2A P29274 1/20 0.38
ADORA2B P29275 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20765601 1.00 TGFBR1 (0.43) TGFBR1AAK1CYP3A4PIK3C3TGFBR2
SCHEMBL20782235 0.93 DHODH (0.38) TGFBR1AAK1CYP3A4PIK3C3
SCHEMBL20765639 0.92 AAK1 (0.43) AAK1CYP3A4PIK3C3
SCHEMBL30514775 0.92 AAK1 (0.43) AAK1CYP3A4PIK3C3
SCHEMBL20765313 0.88 PIK3C3 (0.48) TGFBR1AAK1CYP3A4PIK3C3ADORA3
SCHEMBL30514769 0.88 PIK3C3 (0.48) TGFBR1AAK1CYP3A4PIK3C3ADORA3
SCHEMBL30514770 0.88 PIK3C3 (0.46) TGFBR1AAK1CYP3A4PIK3C3TGFBR2
SCHEMBL20782477 0.88 PIK3C3 (0.46) TGFBR1AAK1CYP3A4PIK3C3TGFBR2
SCHEMBL20764792 0.83 AAK1 (0.49) TGFBR1AAK1CYP3A4PIK3C3
SCHEMBL20776135 0.83 PIK3C3 (0.41) PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116903526-A Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-10-20 CN disclosed
CN-116891431-A Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-10-17 CN disclosed
CN-111094244-B Pyridinylpyridinone compounds 思普瑞特生物科学公司 2023-07-11 CN disclosed