SCHEMBL30522697

SCHEMBL30522697

Cn1c(C2(O)CC2)nc2c1CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAPT P10636 3/20 0.40
ESR2 Q92731 1/20 0.39
ADORA1 P30542 2/20 0.39
NR1H2 P55055 1/20 0.39
PARP1 P09874 1/20 0.38
TNKS2 Q9H2K2 1/20 0.38
PARP2 Q9UGN5 1/20 0.38
MAP3K14 Q99558 1/20 0.38
DDB1 Q16531 3/20 0.37
CRBN Q96SW2 3/20 0.37
GRAMD1A Q96CP6 1/20 0.37
CNR2 P34972 1/20 0.36
P2RX3 P56373 1/20 0.35
HPGDS O60760 1/20 0.35
KDM4E B2RXH2 1/20 0.34
USP2 O75604 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17949105 0.83 MAPT (0.42) MAPTESR2ADORA1NR1H2PARP1
SCHEMBL28477398 0.82 CNR2 (0.32) CNR2
SCHEMBL23632994 0.81 MAPT (0.43) MAPTESR2ADORA1NR1H2PARP1
SCHEMBL28881468 0.81 MAPT (0.46) MAPTESR2ADORA1NR1H2PARP1
SCHEMBL29191201 0.79 ADORA1 (0.46) MAPTESR2ADORA1NR1H2PARP1
SCHEMBL20323953 0.78 PARP1 (0.41) MAPTESR2ADORA1NR1H2PARP1
SCHEMBL22675497 0.78 ADORA1 (0.46) MAPTESR2ADORA1NR1H2PARP1
SCHEMBL5646141 0.78 DPP4 (0.47) MAPTESR2ADORA1NR1H2PARP1
SCHEMBL19713029 0.77 NR1H2 (0.44) MAPTESR2ADORA1NR1H2PARP1
SCHEMBL30522679 0.74 PARP1 (0.37) MAPTESR2NR1H2PARP1TNKS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111925367-B Fused ring derivative inhibitor, preparation method and application thereof 上海翰森生物医药科技有限公司 2023-07-07 CN disclosed